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Medicinal Chemistry
Published by Bentham Science Publishers Ltd..
ISSN 1573-4064
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Aims & scope
Medicinal Chemistry publishes peer-reviewed research. Manuscripts pass a technical check and a scope check by the handling editor before going to independent reviewers.
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Recently published
Development of Pyrazole and Pyrazolo[4,5-b]pyridine Analogues with Potent Fungal Biofilm Inhibition Properties
DOI 10.2174/0115734064519687260917115009 Mohammed Al-Ghorbani, Khulud M. Al-Taisan, Mohammed Baashen, Lakshmi Jayaram, Ramith Ramu · 2026
Organotin (IV)–4-(2-Thienyl) Butyric Acid Complexes Synergize with Vitamins D and E to Inhibit Breast Cancer Cell Proliferation
DOI 10.2174/0115734064509559260927160057 Syeda Saba Shah, Balquees Kanwal, Yasmeen Cheema, Warda Gul, Farzana Shaheen, Rumeza Hanif · 2026
Design, Discovery, Synthesis, Molecular Docking, MD Simulation, and In Vitro Biological Evaluation of Thiazolidinedione-Clubbed Benzimidazole Hybrids as Potential Anticancer Agents
DOI 10.2174/0115734064490624260925075551 Pragya Dubey, DharamPal Pathak, Archana Sharma, Satyam Sharma, Garima Chauhan, Md Azhar Iqbal, Rajeev Taliyan, Shobha Kumari · 2026
Pyrazinone Derivatives in Medicinal Chemistry: SAR Insights and Emerging Therapeutic Applications
DOI 10.2174/0115734064519985260907100959 Neetu Agrawal, Priya Kushwah, Shilpi Pathak · 2026
Nitrogen-Containing Heterocycles in Antibacterial Drug Discovery: Recent Advances and Structure-Activity Relationships
DOI 10.2174/0115734064511285260901071524 Xiaoqing Zhu, Ping Zhang, Xueyu Wang, Meiran Jiao, Hui Sun, Bin Cui · 2026
Computer-Aided Design of Novel Acrylamido Derivatives as Potential Oral Antidiabetic Agents
DOI 10.2174/0115734064513164260828103027 Ahmet Mesut Şentürk, Abdulilah Ece, Süreyya Ölgen · 2026
Uracil-Quinazoline Hybrids: Cytotoxicity, Docking, MD, and DFT Studies
DOI 10.2174/0115734064514052260819104552 Mahkameh Moradimehrabadi, Sara Sadeghian, Alireza Poustforoosh, Leila Emami, soghra khabnadideh · 2026
Pyrimidine Derivatives as Anticancer Agents: Structural Insights and SAR
Studies
DOI 10.2174/0115734064503567260817161010 Balasubramanian Narasimhan, Ashu Sapra · 2026
Arylsulfonylaminopyridines as Potential Epac Inhibitors: Design, Synthesis and Effects on Myocardial Strips
DOI 10.2174/0115734064504072260724092027 Tatiana Vorobeva, Grigory Mokrov, Valeriy Stolyaruk, Daniel Malikin, Andrey Pantileev, Alexey Rebeko, Anna Maksimenko, Iosif Tsorin, Sergey Kryzhanovskii, Vladimir Dorofeev · 2026
From Docking Scores to Biological Relevance: Strengthening Experimental Validation in Medicinal Chemistry Research
DOI 10.2174/0115734064521007260729061037 Vipan Kumar · 2026
Histone Deacetylase (HDAC) Inhibitors: Research and Therapeutic Applications in Cancer and Neurodegenerative Diseases: A Mini-review
DOI 10.2174/0115734064505531260713070531 Yupeng Wu, Siyi Wu, Xin Wang, Hui Sun, Bin Cui · 2026
Drug Repurposing against the PurS Subunit of Phosphoribosylformylglycinamidine Synthase in Methicillin- and Oxacillin-Resistant Staphylococcus Aureus: In vitro and In silico Studies
DOI 10.2174/0115734064472830260611114241 Faryal Ashraf, M. Iqbal Choudhary, Muhammad Yousuf, Humaira Zafar, Atia-tul-Wahab · 2026
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